Abstract
A new series of morpholine derivatives has been identified as selective DA D3 receptor antagonists; their in vitro profile and pharmacokinetic data are provided.
Keywords:
7-TM; Antagonist; DA D3 receptor; Dopamine; Morpholine.
Copyright © 2016 Elsevier Ltd. All rights reserved.
MeSH terms
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Animals
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Binding Sites
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Dopamine D2 Receptor Antagonists / chemical synthesis
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Dopamine D2 Receptor Antagonists / chemistry*
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Dopamine D2 Receptor Antagonists / pharmacokinetics
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Half-Life
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Molecular Docking Simulation
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Morpholines / chemical synthesis
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Morpholines / chemistry*
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Morpholines / pharmacokinetics
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Protein Structure, Tertiary
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Rats
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Receptors, Dopamine D3 / antagonists & inhibitors*
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Receptors, Dopamine D3 / metabolism
Substances
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Dopamine D2 Receptor Antagonists
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Morpholines
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Receptors, Dopamine D3
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morpholine